SCHEMBL8197166

SCHEMBL8197166

c1ccc(-c2ccc(C3CC(c4ccc(C5=NCCN5)cc4)=NO3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 9/20 0.60
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
HPGD P15428 1/20 0.52
CASP1 P29466 1/20 0.52
CASP7 P55210 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MAOB P27338 1/20 0.49
GAA P10253 1/20 0.46
TSHR P16473 1/20 0.46
TOP2A P11388 2/20 0.43
TOP2B Q02880 2/20 0.43
LMNA P02545 1/20 0.41
RECQL P46063 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195231 0.95 NISCH (0.55) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8200553 0.88 NISCH (0.60) NISCHMAOBTOP2ATOP2BLMNA
SCHEMBL8219724 0.88 TOP2A (0.43) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8187010 0.88 LMNA (0.58) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8190284 0.88 ATM (0.44) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8196690 0.86 RARA (0.45) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8187862 0.86 NISCH (0.56) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8516438 0.84 FDPS (0.50) NISCHALDH1A1
SCHEMBL8197475 0.81 MAOB (0.49) NISCHALDH1A1CYP1A2HPGDCASP1
SCHEMBL8195501 0.81 NISCH (0.53) NISCHALDH1A1CYP1A2HPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000078726-A1 IMIDAZOLINE DERIVATIVES FOR THE TREATMENT OF DIABETES, ESPECIALLY TYPE II DIABETES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed