SCHEMBL8198112

SCHEMBL8198112

C=C(OCC)c1nc2sc(Cc3ccccc3)cc2c(=O)[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
ALDH1A1 P00352 4/20 0.43
NPC1 O15118 2/20 0.43
MAPT P10636 2/20 0.43
RAB9A P51151 2/20 0.43
LMNA P02545 1/20 0.43
AGTR1 P30556 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ADORA1 P30542 9/20 0.41
ADORA2A P29274 7/20 0.41
TMIGD3 P0DMS9 2/20 0.41
KDM4E B2RXH2 2/20 0.40
BRD4 O60885 1/20 0.40
PDE5A O76074 1/20 0.39
HPGD P15428 2/20 0.39
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188233 0.89 ALDH1A1 (0.51) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL8203016 0.85 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL8198855 0.83 RAB9A (0.61) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL8190700 0.82 PDE5A (0.47) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL8195845 0.77 ALDH1A1 (0.40) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL31716664 0.75 TNKS2 (0.53) ALDH1A1MAPTKDM4EBRD4HPGD
SCHEMBL8200741 0.75 TNKS2 (0.53) ALDH1A1MAPTKDM4EBRD4HPGD
SCHEMBL8195380 0.75 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL7058912 0.75 SMN1; SMN2 (0.74) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL8200644 0.75 ALDH1A1 (0.57) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063668-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-05-29 WO disclosed