SCHEMBL8198322

SCHEMBL8198322

O=C(c1cccc(Cl)c1)c1ccc(C(F)(F)F)nc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PARP1 P09874 1/20 0.42
ALOX15 P16050 1/20 0.42
CNR2 P34972 1/20 0.42
GRM5 P41594 2/20 0.42
LTC4S Q16873 1/20 0.41
CNR1 P21554 1/20 0.41
GAA P10253 1/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4D Q08499 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ERCC5 P28715 1/20 0.40
FEN1 P39748 1/20 0.40
BDKRB1 P46663 1/20 0.40
FLT1 P17948 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195937 0.86 MAPT (0.41) MAPTKMT2APARP1CNR2LTC4S
SCHEMBL1513035 0.85 GLA (0.44) LMNAMAPTKMT2ACNR2GAA
SCHEMBL6220889 0.82 GRM5 (0.50) KMT2APARP1ALOX15GRM5ALDH1A1
SCHEMBL8196200 0.81 MAPT (0.40) LMNAMAPTKMT2ASMN1; SMN2GRM5
SCHEMBL8194190 0.79 ALDH1A1 (0.49) MAPTPARP1ALOX15GRM5ALDH1A1
SCHEMBL15647834 0.77 GRM5 (0.52) LMNAMAPTKMT2ASMN1; SMN2GRM5
SCHEMBL8198559 0.77 CYP3A4 (0.44) PARP1ALOX15CYP3A4CYP2C19PDE4B
SCHEMBL16632079 0.75 VNN1 (0.48) LMNAMAPTKMT2ASMN1; SMN2PARP1
SCHEMBL165279 0.75 KEAP1 (0.46) LMNASMN1; SMN2ALDH1A1
SCHEMBL30489829 0.75 SMO (0.39) LMNAGAAPDE4BPDE4DFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136810-A DRUGS AS ENZYME INHIBITORS OF PHOSPHODIESTERASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0885894-A1 PYRIDO [2,3-D] PYRIMIDINE DERIVATIVES AND MEDICINAL COMPOSITIONS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-23 EP disclosed