SCHEMBL8199129

SCHEMBL8199129

COc1cc(O)cc(C=Cc2ccc(N(c3ccc(C)cc3)c3ccc(C)cc3)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.67
ALOX5 P09917 5/20 0.67
CYP1A1 P04798 4/20 0.67
CYP1B1 Q16678 4/20 0.67
TTR P02766 3/20 0.67
KDM4E B2RXH2 3/20 0.60
MEN1 O00255 2/20 0.60
MAPT P10636 2/20 0.60
KMT2A Q03164 2/20 0.60
USP2 O75604 1/20 0.60
ALDH1A1 P00352 1/20 0.60
TP53 P04637 1/20 0.60
CYP3A4 P08684 1/20 0.60
HPGD P15428 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
TRPV1 Q8NER1 1/20 0.60
HSD17B10 Q99714 1/20 0.60
PTGS1 P23219 4/20 0.59
NQO2 P16083 4/20 0.59
ABL1 P00519 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199126 1.00 PTGS2 (0.67) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL8206188 0.91 CYP1A1 (0.62) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL8206185 0.91 CYP1A1 (0.62) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL12729821 0.91 PTGS2 (0.80) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL8205829 0.88 PTGS1 (0.66) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL8205830 0.88 PTGS1 (0.66) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL10126425 0.85 RELA (0.66) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL16168068 0.84 CYP1A1 (0.71) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL16167739 0.83 CYP1A1 (0.61) PTGS2ALOX5CYP1A1CYP1B1TTR
SCHEMBL7904563 0.82 RELA (0.78) PTGS2ALOX5CYP1A1CYP1B1TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6066757-A MAY BE INCORPORATED INTO PHOTOCONDUCTING LAYER OF ELECTROPHOTOGRAPHIC PHOTOCONDUCTOR AS CHARGE TRANSPORTING MATERIAL RICOH COMPANY, LTD. (JP) 2000-05-23 US disclosed
US-5641598-A HAVING HIGH RESISTANCE TO THERMAL AND MECHANICAL SHOCK RICOH COMPANY, LTD. (JP) 1997-06-24 US disclosed