Glucuronate

Glucuronate

SCHEMBL8199162

O=C(O)[C@H]1OC(O)[C@H](O)[C@@H](O)[C@@H]1O.Sc1ncnc2nc[nH]c12

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPAT

The experimentally established mechanism targets of Glucuronate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
LMNA P02545 3/20 0.35
HTT P42858 2/20 0.35
TOP2A P11388 2/20 0.35
BRAF P15056 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 1/20 0.34
PI4KA P42356 2/20 0.34
PI4K2B Q8TCG2 2/20 0.34
PI4K2A Q9BTU6 2/20 0.34
PI4KB Q9UBF8 2/20 0.34
DRD3 P35462 1/20 0.34
XDH P47989 1/20 0.34
LRRK2 Q5S007 1/20 0.34
CYP1A2 P05177 2/20 0.34
HIF1A Q16665 2/20 0.34
CDK2 P24941 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mercaptopurine Anhydrous SCHEMBL905281 0.81 HTT (0.37) LMNAHTTTSHRPI4KAPI4K2B
Mercaptopurine Anhydrous SCHEMBL4456159 0.80 HTT (0.38) LMNAHTTTSHRPI4KAPI4K2B
Ribose (Furanose) SCHEMBL831005 0.79 CYP3A4 (0.39) LMNAHTTTSHRPI4KAPI4K2B
Ribose (Furanose) SCHEMBL7680729 0.79 CYP3A4 (0.39) LMNAHTTTSHRPI4KAPI4K2B
Mercaptopurine Anhydrous SCHEMBL29684795 0.73 LMNA (0.57) LMNAHTTPI4KAPI4K2BPI4K2A
Mercaptopurine Anhydrous SCHEMBL8844 0.73 LMNA (0.57) LMNAHTTPI4KAPI4K2BPI4K2A
Mercaptopurine Anhydrous SCHEMBL734088 0.72 LMNA (0.55) LMNAHTTPI4KAPI4K2BPI4K2A
Mercaptopurine Anhydrous SCHEMBL30834915 0.72 LMNA (0.55) LMNAHTTPI4KAPI4K2BPI4K2A
Mercaptopurine Anhydrous SCHEMBL31379732 0.72 LMNA (0.55) LMNAHTTPI4KAPI4K2BPI4K2A
Mercaptopurine Anhydrous SCHEMBL5144254 0.72 LMNA (0.55) LMNAHTTPI4KAPI4K2BPI4K2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6146658-A ADMINISTERING A GLYCOSYL-SPACER-DRUG COMPOUND WHERE THE GLYCOSYL IS A SACCHARIDE WHICH CAN BE ENZYMATICALLY CLEAVED; DRUG IS ANTIINFLAMMATORY, IMMUNOSUPPRESSIVE OR ANTITUMOR AGENT WHICH HYDROXYL OR AMINO GROUP; SELF-ELIMINATING SPACER HOECHST AKTIENGESELLSCHAFT (DE) 2000-11-14 US disclosed
US-5955100-A TREATMENT OF MALIGNANT TUMORS, INFLAMMATORY DISEASES, OR AUTOIMMUNE DISEASES BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1999-09-21 US disclosed