SCHEMBL8199933

SCHEMBL8199933

CSc1ccc(-c2[nH]nc(Cl)c2-c2ccc(Cl)c(C)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.37
MAP4K1 Q92918 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
EIF2AK1 Q9BQI3 1/20 0.33
GSK3B P49841 3/20 0.33
GCGR P47871 2/20 0.32
MAPK14 Q16539 2/20 0.32
STK10 O94804 1/20 0.32
CLK2 P49760 1/20 0.32
GSK3A P49840 1/20 0.32
SLK Q9H2G2 1/20 0.32
CCNE2 O96020 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
PTGS2 P35354 2/20 0.31
GABRP O00591 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8187489 0.83 MAPT (0.39) MAP4K1GSK3BMAPK14CCNE2CDK4
SCHEMBL8642444 0.81 GSK3B (0.45) IKBKBTRPM8GSK3BMAPK14
SCHEMBL8196909 0.79 IKBKB (0.43) IKBKBMAP4K1GSK3BGCGRMAPK14
SCHEMBL8639382 0.79 MAPK14 (0.44) GSK3BGCGRMAPK14GSK3ASLK
SCHEMBL8197292 0.73 PTGS2 (0.40) IKBKBPTGS2PTGS1
SCHEMBL8196899 0.72 PTGS2 (0.39) PTGS2PTGS1
SCHEMBL8188373 0.69 KDM4E (0.48) IKBKBMAP4K1MAPK14
SCHEMBL8069284 0.68 PTGS2 (0.53) MAP4K1PTGS2PTGS1
SCHEMBL6886003 0.68 HSD17B10 (0.41)
SCHEMBL8195709 0.66 GSK3B (0.41) GSK3BMAPK14CLK2CDK2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed