SCHEMBL8196899

SCHEMBL8196899

Cc1cc(-c2c(Cl)n[nH]c2-c2ccc(S(=O)(=O)CCCO)cc2)ccc1Cl

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.39
CA2 P00918 2/20 0.39
PTGS1 P23219 3/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
BRD4 O60885 1/20 0.36
BRD2 P25440 1/20 0.36
BRD3 Q15059 1/20 0.36
SRC P12931 4/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
FFAR1 O14842 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
ABL1 P00519 1/20 0.32
PDGFRB P09619 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8197292 0.94 PTGS2 (0.40) PTGS2CA2PTGS1PTGDR2BRD4
SCHEMBL8200031 0.92 PTGS2 (0.39) PTGS2CA2PTGS1PTGDR2BRD4
SCHEMBL8188503 0.90 PTGS2 (0.40) PTGS2CA2PTGS1PTGDR2NR1H2
SCHEMBL8196142 0.88 PTGS2 (0.37) PTGS2CA2PTGS1PTGDR2BRD4
SCHEMBL8196062 0.87 ALDH1A1 (0.46) PTGS2CA2ALDH1A1CYP3A4CYP2C9
SCHEMBL8196014 0.87 ALDH1A1 (0.37) PTGS2CA2PTGDR2ALDH1A1
SCHEMBL8199737 0.85 PTGS2 (0.40) PTGS2CA2PTGS1PTGDR2BRD4
SCHEMBL8188096 0.85 PTGS2 (0.42) PTGS2PTGS1PTGDR2
SCHEMBL8196010 0.84 CA2 (0.43) PTGS2CA2PTGS1PTGDR2
SCHEMBL8196195 0.84 PTGS2 (0.40) PTGS2CA2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed