SCHEMBL8200071

SCHEMBL8200071

O=C(O)N1Cc2cnc(O)cc2C1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.34
HSP90AA1 P07900 7/20 0.33
HSP90AB1 P08238 4/20 0.32
HSP90B1 P14625 2/20 0.32
TRAP1 Q12931 1/20 0.32
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5316006 0.86 ESR2 (0.39) HSP90AA1HSP90AB1ESR1ESR2
SCHEMBL22445538 0.80 KDM4E (0.41) NAMPT
SCHEMBL29084829 0.76 HDAC1 (0.49) NAMPTESR2HDAC1
SCHEMBL30585116 0.76 HDAC1 (0.49) NAMPTESR2HDAC1
SCHEMBL23856225 0.75 NOTUM (0.53) HSP90AA1HSP90AB1ESR1ESR2
SCHEMBL30063573 0.75 NOTUM (0.53) HSP90AA1HSP90AB1ESR1ESR2
SCHEMBL28892710 0.75 SLC6A9 (0.36) NAMPT
SCHEMBL8203715 0.74 HTR3A (0.48) HSP90AA1HDAC2
SCHEMBL8195601 0.73 KMO (0.51) NAMPT
SCHEMBL23856219 0.73 KEAP1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033389-A2 MACROCYCLIC HCV INHIBITORS AND THEIR USES NOVARTIS AG (CH) 2008-03-20 WO disclosed