SCHEMBL8200375

SCHEMBL8200375

CCCc1cc(C(=O)NC(Cc2ccccc2)C2=COCO2)c(NC(=O)c2ccc(C(=O)OC)cc2)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
KDM4E B2RXH2 7/20 0.41
HPGD P15428 7/20 0.41
MAPT P10636 8/20 0.40
HSD17B10 Q99714 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
GRIN2C Q14957 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MAPK1 P28482 2/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199938 0.96 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8200396 0.94 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8206226 0.93 ALDH1A1 (0.42) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8210397 0.89 KDM4E (0.41) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8212434 0.89 SMN1; SMN2 (0.39) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL8206045 0.89 GRIN2C (0.39) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL8198895 0.88 SMN1; SMN2 (0.38) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL8207755 0.86 GRIN2C (0.48) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL8212891 0.82 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDMAPTHSD17B10
SCHEMBL8212479 0.81 MAPT (0.38) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed