SCHEMBL8200487

SCHEMBL8200487

COc1ccc(CCCC(=O)c2ccc(OC)cc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.71
RAB9A P51151 2/20 0.71
PDE4B Q07343 1/20 0.68
ALOX5 P09917 1/20 0.64
HDAC8 Q9BY41 3/20 0.60
HDAC1 Q13547 3/20 0.60
MAPT P10636 3/20 0.60
F2RL1 P55085 1/20 0.57
LMNA P02545 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
MMP1 P03956 1/20 0.57
CALM1 P0DP23 1/20 0.56
GSK3B P49841 1/20 0.56
CASP3 P42574 1/20 0.56
SENP8 Q96LD8 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
SENP6 Q9GZR1 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
HDAC3 O15379 1/20 0.56
HDAC4 P56524 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1303471 0.92 NPC1 (0.85) NPC1RAB9APDE4BALOX5HDAC8
SCHEMBL7868896 0.91 NPC1 (0.83) NPC1RAB9APDE4BHDAC8HDAC1
SCHEMBL11776953 0.87 NPC1 (0.82) NPC1RAB9APDE4BALOX5HDAC8
SCHEMBL4082864 0.87 PDE4B (0.86) NPC1RAB9APDE4BHDAC8HDAC1
SCHEMBL3171960 0.87 PDE4B (0.79) NPC1RAB9APDE4BHDAC8HDAC1
SCHEMBL8984314 0.86 THRA (0.67) NPC1RAB9APDE4B
SCHEMBL28650786 0.85 LMNA (0.76) NPC1RAB9APDE4BHDAC8HDAC1
SCHEMBL11436374 0.85 NPC1 (0.73) NPC1RAB9APDE4BMAPTF2RL1
SCHEMBL9151000 0.85 NPC1 (0.64) NPC1RAB9APDE4BALOX5HDAC8
SCHEMBL4096780 0.83 NPC1 (0.71) NPC1RAB9APDE4BHDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840606-B1 DI- AND TRIVALENT SMALL MOLECULE SELECTIN INHIBITORS TEXAS BIOTECHNOLOGY CORP (US) 2000-06-07 EP disclosed
US-5919768-A COMPOUNDS WHICH INHIBIT BINDING OF SELECTINS TO SIALYL-LEWIS-X AND SIALYL-LEWIS-A CARBOHYDRATES TEXAS BIOTECHNOLOGY CORPORATION (US) 1999-07-06 US disclosed