SCHEMBL8200656

SCHEMBL8200656

COc1ccc(CCNC(=O)c2ccc3c(c2)CCC(CCN2CCC(c4ccccc4)CC2)C3=O)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.53
LMNA P02545 2/20 0.53
MAPT P10636 8/20 0.52
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
POLB P06746 2/20 0.46
HTR2C P28335 1/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198570 0.89 HTR2C (0.47) SMN1; SMN2MAPTHTR2CALDH1A1
SCHEMBL8199695 0.88 SLC6A2 (0.46) HTR2C
SCHEMBL8202264 0.87 CHRM4 (0.50) SMN1; SMN2HTR2C
SCHEMBL8191651 0.87 MCHR1 (0.48) SMN1; SMN2LMNAMAPTNPC1RAB9A
SCHEMBL8200603 0.86 HTR2C (0.49) SMN1; SMN2HTR2CALDH1A1
SCHEMBL8588802 0.85 HTR2C (0.48) LMNAMAPTHTR2C
SCHEMBL8198781 0.84 HTR2C (0.46) HTR2CALDH1A1
SCHEMBL8203525 0.84 SIGMAR1 (0.46) HTR2CALDH1A1
SCHEMBL8191618 0.83 HTR2C (0.50) MAPTPOLBHTR2CALDH1A1
SCHEMBL8199972 0.83 HTR2C (0.46) HTR2CGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed