SCHEMBL8198570

SCHEMBL8198570

O=C(NCCc1ccccc1)c1ccc2c(c1)CCC(CCN1CCC(c3ccccc3)CC1)C2=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SLC5A7 Q9GZV3 1/20 0.45
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
MAPT P10636 2/20 0.43
DRD2 P14416 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
CHRM4 P08173 1/20 0.43
SIGMAR1 Q99720 2/20 0.42
HTR2A P28223 1/20 0.42
HTR2B P41595 1/20 0.42
DRD4 P21917 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198781 0.95 HTR2C (0.46) HTR2CDRD2ALDH1A1GLACHRM4
SCHEMBL8191651 0.94 MCHR1 (0.48) HTR2CSMN1; SMN2SLC5A7OPRM1OPRK1
SCHEMBL8203525 0.94 SIGMAR1 (0.46) HTR2CALDH1A1GLACHRM4SIGMAR1
SCHEMBL8202264 0.93 CHRM4 (0.50) HTR2CSMN1; SMN2SLC5A7OPRM1OPRK1
SCHEMBL8200603 0.93 HTR2C (0.49) HTR2CSMN1; SMN2SLC5A7DRD2ALDH1A1
SCHEMBL8199695 0.92 SLC6A2 (0.46) HTR2COPRM1OPRK1DRD2DRD4
SCHEMBL8199804 0.91 HTR2C (0.49) HTR2COPRM1OPRK1DRD2ALDH1A1
SCHEMBL8588802 0.90 HTR2C (0.48) HTR2CSLC5A7OPRM1OPRK1MAPT
SCHEMBL8199074 0.89 HTR2C (0.48) HTR2CSMN1; SMN2OPRM1OPRK1DRD2
SCHEMBL8200656 0.89 SMN1; SMN2 (0.53) HTR2CSMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed