SCHEMBL8201063

SCHEMBL8201063

COC(=O)Cc1cccc(-c2cc(CCCCc3ccc(O)c(-c4cccc(CC(=O)OC)c4)c3)ccc2O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
GAA P10253 1/20 0.51
GFER P55789 1/20 0.51
SLC7A5 Q01650 1/20 0.43
BACE1 P56817 1/20 0.43
CYP4F2 P78329 2/20 0.42
CYP4A11 Q02928 2/20 0.42
ALOX5 P09917 3/20 0.42
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
YWHAG P61981 1/20 0.42
SELP P16109 3/20 0.41
SELPLG Q14242 1/20 0.41
GABRA1 P14867 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6553321 0.99 ALDH1A1 (0.50) ALDH1A1GAAGFERSLC7A5BACE1
SCHEMBL8709712 0.94 ALDH1A1 (0.48) ALDH1A1GAAGFERSLC7A5BACE1
SCHEMBL8200563 0.87 ALDH1A1 (0.51) ALDH1A1GAAGFERSLC7A5CYP4F2
SCHEMBL2589280 0.86 PPARA (0.48) BACE1CYP4F2CYP4A11ALOX5NPC1
SCHEMBL8200129 0.86 JAK2 (0.49) SLC7A5CYP4F2CYP4A11HPGDSELP
SCHEMBL9202609 0.84 ALDH1A1 (0.59) ALDH1A1GAAGFERSLC7A5BACE1
SCHEMBL7035349 0.82 ALDH1A1 (0.50) ALDH1A1GAAGFERSLC7A5CYP4F2
SCHEMBL8200551 0.82 PPARA (0.44) CYP4F2CYP4A11ALOX5NPC1PKM
SCHEMBL14768426 0.80 GAA (0.70) ALDH1A1GAAGFERSLC7A5CYP4F2
SCHEMBL7725121 0.79 BACE1 (0.55) BACE1ALOX5HPGDTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840606-B1 DI- AND TRIVALENT SMALL MOLECULE SELECTIN INHIBITORS TEXAS BIOTECHNOLOGY CORP (US) 2000-06-07 EP disclosed
US-5919768-A COMPOUNDS WHICH INHIBIT BINDING OF SELECTINS TO SIALYL-LEWIS-X AND SIALYL-LEWIS-A CARBOHYDRATES TEXAS BIOTECHNOLOGY CORPORATION (US) 1999-07-06 US disclosed