SCHEMBL8228161

SCHEMBL8228161

CC(=O)OCCSc1ccc(-c2[nH]nc(C(F)(F)F)c2-c2ccc(C)c(Cl)c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 11/20 0.35
PPARA Q07869 7/20 0.35
PPARG P37231 4/20 0.35
CHUK O15111 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NOTUM Q6P988 1/20 0.32
DHODH Q02127 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196758 0.77 MEN1 (0.33) ALDH1A1MEN1KMT2ASMN1; SMN2CYP1A2
SCHEMBL8195825 0.74 PTGS2 (0.38) ALDH1A1MEN1KMT2ASMN1; SMN2PTGS1
SCHEMBL8194817 0.74 PTGS2 (0.40) CHUKALDH1A1PTGS1PTGS2
SCHEMBL8187466 0.73 PTGS2 (0.39) ALDH1A1MEN1KMT2ASMN1; SMN2PTGS1
SCHEMBL8187488 0.73 GRK6 (0.33) ALDH1A1MEN1KMT2ASMN1; SMN2CYP1A2
SCHEMBL8187508 0.73 MEN1 (0.33) MEN1KMT2ASMN1; SMN2CYP1A2CYP2C9
SCHEMBL8202136 0.73 PTGS2 (0.37) CHUKALDH1A1NOTUMPTGS1PTGS2
SCHEMBL8195777 0.73 PTGS2 (0.37) ALDH1A1MEN1KMT2ASMN1; SMN2PTGS1
SCHEMBL8196136 0.71 PTGS2 (0.38) SMN1; SMN2PTGS1PTGS2
SCHEMBL8196086 0.69 ALDH1A1 (0.39) ALDH1A1MEN1KMT2ASMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed