SCHEMBL8202791

SCHEMBL8202791

O=C1c2ccc(OCc3ccccc3)cc2CCC1CN1CCCCC1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.58
MAOB P27338 2/20 0.58
SIGMAR1 Q99720 3/20 0.55
HTR1A P08908 2/20 0.55
HRH3 Q9Y5N1 5/20 0.54
CYP2D6 P10635 3/20 0.54
HRH1 P35367 1/20 0.54
ITGB3 P05106 1/20 0.52
ITGA2B P08514 1/20 0.52
BACE1 P56817 1/20 0.49
METAP1 P53582 2/20 0.49
CYP24A1 Q07973 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8203429 0.90 MAOB (0.59) MAOAMAOBSIGMAR1HTR1AHRH3
SCHEMBL6491492 0.89 ADRA1D (0.54) MAOAMAOBSIGMAR1HTR1AHRH3
SCHEMBL7297935 0.85 ITGB3 (0.49) MAOAMAOBSIGMAR1HTR1AHRH3
SCHEMBL7289032 0.85 ITGB3 (0.49) MAOAMAOBSIGMAR1HTR1AHRH3
SCHEMBL8200894 0.84 ITGB3 (0.58) MAOAMAOBHRH3CYP2D6ITGB3
SCHEMBL29092251 0.81 MAOB (0.58) MAOAMAOBHRH3CYP2D6ITGB3
Hydrochloric Acid SCHEMBL4623367 0.81 CYP24A1 (0.57) SIGMAR1METAP1CYP24A1
SCHEMBL7298191 0.81 ITGB3 (0.47) MAOAMAOBSIGMAR1HTR1AHRH3
SCHEMBL7298201 0.81 ITGB3 (0.47) MAOAMAOBSIGMAR1HTR1AHRH3
SCHEMBL5904289 0.81 CYP24A1 (0.59) SIGMAR1METAP1CYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO disclosed