SCHEMBL8203429

SCHEMBL8203429

O=C1c2ccc(OCCc3ccccc3)cc2CCC1CN1CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.59
MAOA P21397 2/20 0.59
SIGMAR1 Q99720 4/20 0.53
HTR1A P08908 2/20 0.53
CYP24A1 Q07973 1/20 0.52
HRH3 Q9Y5N1 4/20 0.49
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
METAP1 P53582 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202791 0.90 MAOA (0.58) MAOBMAOASIGMAR1HTR1ACYP24A1
SCHEMBL6503237 0.89 SIGMAR1 (0.51) MAOBMAOASIGMAR1HTR1ACYP24A1
Hydrochloric Acid SCHEMBL4623367 0.79 CYP24A1 (0.57) SIGMAR1CYP24A1DRD2HTR2AHTR2C
SCHEMBL5904289 0.79 CYP24A1 (0.59) SIGMAR1CYP24A1DRD2HTR2AHTR2C
SCHEMBL6491492 0.79 ADRA1D (0.54) MAOBMAOASIGMAR1HTR1ACYP24A1
SCHEMBL30423421 0.76 METAP1 (0.74) SIGMAR1HTR1ADRD2HTR2AHTR2C
SCHEMBL7289032 0.76 ITGB3 (0.49) MAOBMAOASIGMAR1HTR1ACYP24A1
SCHEMBL7297935 0.76 ITGB3 (0.49) MAOBMAOASIGMAR1HTR1ACYP24A1
SCHEMBL15839887 0.75 MAOB (1.00) MAOBMAOA
SCHEMBL11732870 0.75 THRA (0.52) SIGMAR1HTR1ACYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed