SCHEMBL7298201

SCHEMBL7298201

Cc1ccc(CC2(O)CCN(C[C@@H]3CCc4cc(OCc5ccccc5)ccc4C3=O)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
CYP24A1 Q07973 4/20 0.44
CYP26A1 O43174 2/20 0.44
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
MAPT P10636 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
SIGMAR1 Q99720 4/20 0.44
HTR1A P08908 2/20 0.44
CYP2D6 P10635 1/20 0.43
HRH1 P35367 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
DRD2 P14416 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298191 1.00 ITGB3 (0.47) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL7289032 0.95 ITGB3 (0.49) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL7297935 0.95 ITGB3 (0.49) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL7289865 0.82 GRIN1 (0.45) GRIN2DGRIN3BMAPTGRIN1GRIN2A
SCHEMBL27408398 0.81 MMP1 (0.43) GRIN2DGRIN3BMAPTGRIN1GRIN2A
SCHEMBL8202791 0.81 MAOA (0.58) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL6491492 0.79 ADRA1D (0.54) ITGB3ITGA2BMAOAMAOBCYP24A1
Hydrochloric Acid SCHEMBL7289438 0.77 SIGMAR1 (0.46) ITGB3ITGA2BGRIN2BSIGMAR1HTR1A
SCHEMBL7286572 0.77 GRIN1 (0.48) ITGB3ITGA2BGRIN2DGRIN3BMAPT
SCHEMBL7288330 0.76 HRH3 (0.48) MAPTGRIN1GRIN2BCYP2D6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6359138-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2002-03-19 US disclosed
EP-0846683-B1 4-Hydroxy-piperidine derivatives HOFFMANN LA ROCHE (CH) 2001-09-19 EP disclosed
EP-0846683-A1 4-Hydroxy-piperidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-06-10 EP disclosed