SCHEMBL8202811

SCHEMBL8202811

CC(=O)NC(C)(C)Cc1c(C(C2=C(O)C(C)(c3ccc(C)cc3)C2O)c2ccccc2)[nH]c2cc(C)ccc12

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.35
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
EGFR P00533 1/20 0.31
MLKL Q8NB16 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196011 0.98 CYP19A1 (0.34) CYP19A1MTNR1AMTNR1BEGFRMLKL
SCHEMBL8203261 0.88 CYP19A1 (0.34) CYP19A1MTNR1AMTNR1B
SCHEMBL8202857 0.88 CYP19A1 (0.34) CYP19A1MTNR1AMTNR1B
SCHEMBL8208702 0.87 MTNR1A (0.38) CYP19A1MTNR1AMTNR1BEGFRMLKL
SCHEMBL3280434 0.85 CYP19A1 (0.35) CYP19A1MTNR1AMTNR1BEGFRMLKL
SCHEMBL8203579 0.84 MTNR1A (0.38) CYP19A1MTNR1AMTNR1BEGFRMLKL
SCHEMBL3284276 0.83 CYP19A1 (0.34) CYP19A1MTNR1AMTNR1BEGFRMLKL
SCHEMBL3280349 0.81 MTNR1A (0.34) CYP19A1MTNR1AMTNR1B
SCHEMBL8203863 0.81 MLKL (0.42) CYP19A1MLKL
SCHEMBL8195891 0.80 CYP19A1 (0.36) CYP19A1MLKL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008043698-A1 VINYLOGOUS ACIDS DERIVATIVES AS CHYMASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2008-04-17 WO disclosed