SCHEMBL8202867

SCHEMBL8202867

Cc1cc(=O)oc2cc(C(=O)NC(=O)[C@@H]3CCCN3C(=O)CNC(=O)OCc3ccccc3)ccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.47
ALDH1A1 P00352 2/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 2/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FKBP1A P62942 4/20 0.41
MAOA P21397 2/20 0.41
MAOB P27338 3/20 0.41
NPC1 O15118 1/20 0.41
CASP3 P42574 1/20 0.41
RAB9A P51151 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
GFER P55789 1/20 0.41
OPRK1 P41145 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740254 0.88 ALDH1A1 (0.51) PREPALDH1A1GAAHPGDLMNA
SCHEMBL29354123 0.88 ALDH1A1 (0.51) PREPALDH1A1GAAHPGDLMNA
SCHEMBL30377081 0.88 ALDH1A1 (0.51) PREPALDH1A1GAAHPGDLMNA
SCHEMBL4189547 0.85 PREP (0.49) PREPALDH1A1GAAHPGDLMNA
SCHEMBL5264694 0.82 PREP (0.55) PREPALDH1A1LMNAGFERNPSR1
SCHEMBL16162942 0.81 KDM4E (0.45) ALDH1A1GAAMAPTHPGDLMNA
SCHEMBL3364774 0.79 PREP (0.49) PREPALDH1A1FKBP1AGFERNPSR1
SCHEMBL15673353 0.79 ATM (0.51) PREPLMNAPOLBFKBP1A
SCHEMBL24709598 0.77 ALDH1A1 (0.49) PREPALDH1A1HPGDLMNAGFER
SCHEMBL29350880 0.77 FAP (0.42) PREPALDH1A1GAAHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090786-A HALOPYRROLE AMIDATED AMINO ACID USEFUL FOR INHIBITING SERINE PROTEASE ACTIVITY FONDATECH BENELUX N.V. (BE) 2000-07-18 US disclosed
EP-0764151-A2 PURIFICATION OF SERINE PROTEASE AND SYNTHETIC INHIBITORS THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 1997-03-26 EP disclosed
WO-1995034538-A2 PURIFICATION OF SERINE PROTEASES AND SYNTHETIC INHIBITORS THEREOF UNIVERSITAIRE INSTELLING ANTWERPEN (BE) 1995-12-21 WO disclosed