SCHEMBL8202889

SCHEMBL8202889

COC(=O)[C@H](CCCCO)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](I)Cc1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IL1RN P18510 8/20 0.55
ERAP2 Q6P179 8/20 0.55
NPY4R P50391 7/20 0.55
NPY1R P25929 5/20 0.55
ERAP1 Q9NZ08 6/20 0.52
NPY2R P49146 4/20 0.47
NPY5R Q15761 3/20 0.47
TSHR P16473 1/20 0.45
LNPEP Q9UIQ6 1/20 0.44
FOLH1 Q04609 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL930562 0.90 IL1RN (0.57) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL930564 0.90 IL1RN (0.57) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL8203393 0.87 NPY4R (0.47) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL8203303 0.83 CAPN1 (0.62) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL28069215 0.73 ERAP2 (0.60) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL28069213 0.73 ERAP2 (0.60) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL30578432 0.72 LNPEP (0.58) ERAP2NPY4RNPY1RLNPEP
SCHEMBL29275108 0.72 IL1RN (0.59) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL29275103 0.72 IL1RN (0.59) IL1RNERAP2NPY4RNPY1RERAP1
SCHEMBL9073868 0.72 OPRK1 (0.65) NPY4RNPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed