SCHEMBL8203033

SCHEMBL8203033

O=C(Nc1ccccc1)c1cc(Br)c[nH]c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPD1 P10809 1/20 0.56
HSPE1 P61604 1/20 0.56
KDR P35968 1/20 0.55
CFTR P13569 1/20 0.54
F12 P00748 2/20 0.51
NTRK1 P04629 1/20 0.50
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
TDP1 Q9NUW8 1/20 0.49
ALDH1A1 P00352 2/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
HTT P42858 2/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4342778 0.84 HSPD1 (0.55) HSPD1HSPE1CFTRF12KMT2A
SCHEMBL5241258 0.82 ITK (0.54) CFTRNTRK1KMT2AMEN1TDP1
SCHEMBL31265782 0.80 PKM (0.61) HSPD1HSPE1KMT2AMEN1ALDH1A1
SCHEMBL15850171 0.76 ITK (0.67) CFTRKMT2AMEN1ALDH1A1HTT
SCHEMBL4725368 0.75 DYRK1A (0.60) KDRALDH1A1HPGDKDM4EHSD17B10
SCHEMBL9967909 0.74 HSPD1 (0.67) HSPD1HSPE1F12KMT2AMEN1
SCHEMBL3368022 0.74 TYK2 (0.70) CFTRKMT2AMEN1TDP1ALDH1A1
SCHEMBL15837010 0.73 ERCC1 (0.53) KDRKMT2AALDH1A1MAOAMAOB
SCHEMBL23825504 0.73 SORT1 (0.74) HSPD1HSPE1F12ALDH1A1
SCHEMBL29980628 0.73 SORT1 (0.74) HSPD1HSPE1F12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021725-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-21 WO disclosed