SCHEMBL8204830

SCHEMBL8204830

CC1COc2c(F)cccc2O1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.50
CYP19A1 P11511 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.37
CYP11B1 P15538 4/20 0.36
CYP11B2 P19099 4/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
CHRNB4 P30926 3/20 0.35
CHRNA3 P32297 3/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
TERT O14746 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8204827 0.79 CA2 (0.50) CA2CYP19A1L3MBTL1CYP11B1CYP11B2
SCHEMBL8199657 0.79 CHRNB4 (0.54) CA2ADRA1DADRA1AADRA1BCHRNB4
SCHEMBL13998649 0.76 ADRA1D (0.50) CYP19A1ADRA1DADRA1AADRA1BMAPK1
SCHEMBL8125243 0.76 CA2 (0.58) CA2CYP19A1L3MBTL1CYP11B1CYP11B2
SCHEMBL1044198 0.75 PARP1 (0.33)
SCHEMBL7218131 0.75 CA2 (0.47) CA2CYP19A1L3MBTL1CYP11B1CYP11B2
SCHEMBL1519103 0.73 CA2 (0.49) CA2CYP19A1L3MBTL1CYP11B1CYP11B2
SCHEMBL7216342 0.73 CA2 (0.52) CA2L3MBTL1CYP11B1CYP11B2MAPK1
SCHEMBL30499165 0.73 CA2 (0.41) CA2CYP19A1L3MBTL1ADRA1DADRA1A
SCHEMBL266615 0.72 NISCH (0.48) CHRNB4CHRNA3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000058301-A1 N-[2-(4-AMINOPHYL)ETHYL]-2,3-DIHYDRO-1,4-BENZODIOXINE-2-METHANAMINE, PRODUCTION AND THERAPEUTIC USE THEREOF SANOFI-SYNTHELABO (FR) 2000-10-05 WO disclosed