SCHEMBL8207134

SCHEMBL8207134

COCCc1c(C(=O)O)[nH]c(-c2[nH]c(C(=O)O)c(CCOC)c2C(=O)O)c1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.37
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 1/20 0.35
LMNA P02545 1/20 0.34
ALDH1A1 P00352 2/20 0.34
GPR17 Q13304 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MCL1 Q07820 8/20 0.33
BCL2 P10415 3/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8202821 0.76 LMNA (0.44) HCAR2CYP1A2CYP2C9LMNAALDH1A1
SCHEMBL5612429 0.74 HCAR2 (0.40) HCAR2LMNAALDH1A1KDM4EHSD17B10
SCHEMBL9816497 0.70 MCL1 (0.67) ALDH1A1KDM4EHSD17B10MCL1BCL2
SCHEMBL8203697 0.67 HPGD (0.59) LMNAALDH1A1KDM4EHPGD
SCHEMBL28610448 0.67 HCAR2 (0.39) HCAR2CYP2C9LMNAALDH1A1KDM4E
SCHEMBL9955516 0.66 ALDH1A1 (0.46) HCAR2LMNAALDH1A1HPGDHSD17B10
SCHEMBL1126546 0.65 HPGD (0.64) CYP1A2CYP2C9LMNAALDH1A1KDM4E
SCHEMBL17797893 0.64 TSHR (0.46) HCAR2CYP1A2LMNAALDH1A1KDM4E
SCHEMBL5611550 0.64 TSHR (0.34) HCAR2ALDH1A1
SCHEMBL17797824 0.63 TSHR (0.38) HCAR2CYP1A2CYP2C9ALDH1A1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0591355-B1 PORPHYCENE COMPOUNDS FOR PHOTODYNAMIC THERAPY CYTOPHARM INC (US) 2000-03-08 EP disclosed
US-5409900-A Treatment of cancer tumors, psoriasis; purification of blood CYTOPHARM, INC. (US) 1995-04-25 US disclosed
US-5262401-A Porphyrins as antitumor agents and psoriasis treatment CYTOPHARM, INC. (US) 1993-11-16 US disclosed
US-5179120-A Antitumor agents or psoriasis CYTOPHARM, INC. (US) 1993-01-12 US disclosed