SCHEMBL8207485

SCHEMBL8207485

N#Cc1cc(C(=O)N=C(N)N)ccc1Oc1cccnc1

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
CYP19A1 P11511 5/20 0.53
MAPK14 Q16539 1/20 0.44
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
GRM5 P41594 1/20 0.40
AOC3 Q16853 1/20 0.40
SLC22A12 Q96S37 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8179683 0.81 ALDH1A1 (0.61) ALDH1A1SMN1; SMN2CYP19A1MAPK14KDM4E
SCHEMBL8185434 0.80 SLC9A1 (0.52) ALDH1A1SMN1; SMN2KDM4EMEN1GAA
SCHEMBL8172578 0.79 SLC9A1 (0.50)
SCHEMBL8474697 0.79 PTGS1 (0.46) ALDH1A1KDM4EMEN1GAAMAPK1
SCHEMBL8183089 0.78 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2KDM4EMEN1GAA
SCHEMBL8832380 0.78 KDM4E (0.45) ALDH1A1KDM4EMEN1GAAMAPK1
SCHEMBL8170154 0.78 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2KDM4EMEN1GAA
SCHEMBL8177782 0.77 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2CYP19A1
SCHEMBL5565443 0.76 ALDH1A1 (0.73) ALDH1A1SMN1; SMN2CYP19A1MAPK14KDM4E
Hydrochloric Acid SCHEMBL8506934 0.74 ALDH1A1 (0.49) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022883-A Heterocyclyloxybenzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-02-08 US disclosed
EP-0694537-A1 Heterocyclyloxy- benzoylguanidine derivatives, their preparation and their use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GmbH (DE) 1996-01-31 EP disclosed