SCHEMBL8474697

SCHEMBL8474697

CS(=O)(=O)Nc1cc(C(=O)N=C(N)N)ccc1Oc1cccnc1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.46
PTGS2 P35354 4/20 0.46
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
ALPL P05186 1/20 0.41
BRD4 O60885 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8471438 0.85 PTGS1 (0.54) PTGS1PTGS2KDM4EMEN1ALDH1A1
SCHEMBL8172578 0.84 SLC9A1 (0.50)
SCHEMBL8474684 0.83 PTGS1 (0.45) PTGS1PTGS2KDM4EMEN1ALDH1A1
SCHEMBL8832380 0.80 KDM4E (0.45) KDM4EMEN1ALDH1A1GAAMAPK1
SCHEMBL8207485 0.79 ALDH1A1 (0.57) KDM4EMEN1ALDH1A1GAAMAPK1
SCHEMBL8185434 0.77 SLC9A1 (0.52) KDM4EMEN1ALDH1A1GAAMAPK1
SCHEMBL8183089 0.75 SMN1; SMN2 (0.47) KDM4EMEN1ALDH1A1GAAMAPK1
SCHEMBL8170154 0.74 SMN1; SMN2 (0.46) KDM4EMEN1ALDH1A1GAAMAPK1
SCHEMBL8179861 0.74 SLC9A1 (0.56)
SCHEMBL8180285 0.73 SLC9A1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856344-A CARDIOVASCULAR DISORDERS; ANTIARRHYTHMIA AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; STOCK HOECHST AKTIENGESELLSCHAFT (DE) 1999-01-05 US claimed
US-5856344-A CARDIOVASCULAR DISORDERS; ANTIARRHYTHMIA AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; STOCK HOECHST AKTIENGESELLSCHAFT (DE) 1999-01-05 US disclosed
EP-0774459-A1 Sulfonylamino-substituted benzoylguanidines, process for their preparation, their use as medicament or diagnostic agent as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-21 EP disclosed