SCHEMBL8207845

SCHEMBL8207845

COC(=O)C1CCC(C(=O)Nc2sc(Cl)cc2C(=O)NCc2cccc([N+](=O)[O-])c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.47
ACKR3 P25106 1/20 0.44
MAPT P10636 2/20 0.44
POLB P06746 2/20 0.43
PTPN1 P18031 2/20 0.41
ALDH1A1 P00352 3/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
RIPK1 Q13546 1/20 0.39
RIPK3 Q9Y572 1/20 0.39
SENP5 Q96HI0 1/20 0.39
SENP2 Q9HC62 1/20 0.39
SENP1 Q9P0U3 1/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420131 0.91 AKR1B1 (0.48) AKR1B1ACKR3MAPTPOLBPTPN1
SCHEMBL8206201 0.90 MAPT (0.46) AKR1B1ACKR3MAPTPOLBPTPN1
SCHEMBL8206839 0.90 MAPT (0.49) AKR1B1ACKR3MAPTPOLBALDH1A1
Bicarbonate SCHEMBL7420135 0.89 POLB (0.51) AKR1B1ACKR3MAPTPOLBALDH1A1
SCHEMBL8207740 0.87 HPGD (0.42) MAPTPOLBALDH1A1LMNASMN1; SMN2
SCHEMBL7424534 0.83 MAPT (0.47) AKR1B1ACKR3MAPTPOLBALDH1A1
SCHEMBL7430376 0.82 ACKR3 (0.48) AKR1B1ACKR3MAPTPOLBPTPN1
SCHEMBL8207774 0.82 LMNA (0.47) POLBALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL8207562 0.82 ALDH1A1 (0.43) MAPTPOLBALDH1A1LMNAKDM4E
SCHEMBL8207861 0.81 LMNA (0.46) LMNAMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed