SCHEMBL8207740

SCHEMBL8207740

COC(=O)C1CCC(C(=O)Nc2sc(Cl)cc2C(=O)NCc2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.42
GLA P06280 2/20 0.42
TP53 P04637 2/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD11B1 P28845 1/20 0.42
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
HIF1A Q16665 1/20 0.41
NPC1 O15118 2/20 0.41
PKM P14618 2/20 0.41
RAB9A P51151 2/20 0.41
DRD4 P21917 4/20 0.41
DRD3 P35462 1/20 0.41
HSP90AA1 P07900 1/20 0.41
PPARG P37231 2/20 0.41
LMNA P02545 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8207562 0.90 ALDH1A1 (0.43) ALDH1A1MAPTPOLBGAAHIF1A
SCHEMBL8199985 0.90 NPC1 (0.46) TP53ALDH1A1MAPTPOLBGAA
SCHEMBL7892994 0.90 USP2 (0.45) HPGDTP53USP2ALDH1A1HSD11B1
SCHEMBL8207368 0.89 REV1 (0.47) HPGDGLATP53USP2ALDH1A1
SCHEMBL8212725 0.88 GAA (0.56) HPGDGLATP53USP2ALDH1A1
SCHEMBL8207845 0.87 AKR1B1 (0.47) HPGDTP53ALDH1A1MAPTPOLB
Bicarbonate SCHEMBL7892996 0.87 HPGD (0.50) HPGDTP53USP2ALDH1A1MAPT
SCHEMBL8207774 0.87 LMNA (0.47) HPGDALDH1A1POLBNPC1PKM
SCHEMBL8207861 0.86 LMNA (0.46) HPGDGAANPC1PKMRAB9A
SCHEMBL8211919 0.84 KDM4E (0.54) HPGDMAPTPOLBGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed