SCHEMBL8208049

SCHEMBL8208049

C=CCOc1ccc(C[C@H](BOCN)C(=O)N[C@H](C(=O)O)C(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.39
GAA P10253 1/20 0.37
PPARG P37231 2/20 0.36
PPARA Q07869 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ACACB O00763 2/20 0.35
FFAR1 O14842 1/20 0.35
ADAMTS4 O75173 5/20 0.35
CYP2D6 P10635 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MMP13 P45452 1/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195215 0.92 ACACB (0.35) GAAPPARGALDH1A1ACACBFFAR1
SCHEMBL8208453 0.90 ITGB3 (0.36) PPARGITGB3ITGA2BMMP13
SCHEMBL12907630 0.87 NPSR1 (0.40) NPSR1PPARGPPARAALDH1A1ACACB
SCHEMBL8208994 0.87 MME (0.42) ITGB3ITGA2BALDH1A1
SCHEMBL12943110 0.86 CTSD (0.34) GAAACACBCYP2D6MEN1KMT2A
SCHEMBL8209040 0.86 SMN1; SMN2 (0.34) GAAALDH1A1ACACBCYP2D6MEN1
SCHEMBL12943109 0.86 ACACB (0.35) GAAALDH1A1ACACBFFAR1CYP2D6
SCHEMBL8205374 0.84 FFAR1 (0.40) PPARGPPARAITGB3ITGA2BALDH1A1
SCHEMBL12943104 0.83 IL1RN (0.33) PPARG
SCHEMBL8201294 0.83 PTPN1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110021434-A1 Macrocyclic Cysteine Protease Inhibitors and Compositions Thereof UNIVERSITY OF CANTERBURY (NZ) 2011-01-27 US disclosed
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021434-A1 Macrocyclic Cysteine Protease Inhibitors and Compositions Thereof CAPNS1, CAPN1, CAPN9 NPSR1 4228/4885GAA 524/4885PPARG 3703/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.