SCHEMBL8209040

SCHEMBL8209040

C=CCOc1ccc(C[C@H](BOCN)C(=O)N[C@H](C(=O)N[C@H](C=O)CC=C)C(C)C)cc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.34
CTSB P07858 1/20 0.32
ACACB O00763 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
GAA P10253 1/20 0.32
CASP1 P29466 1/20 0.32
CYP2D6 P10635 1/20 0.31
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
ALDH1A1 P00352 1/20 0.31
BMP1 P13497 1/20 0.31
NPC1 O15118 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208453 0.88 ITGB3 (0.36) MMP1MMP2MMP9
SCHEMBL12943214 0.87 CTSB (0.38) SMN1; SMN2CTSBACACBGAACYP2D6
SCHEMBL8208049 0.86 NPSR1 (0.39) SMN1; SMN2ACACBMEN1KMT2AGAA
SCHEMBL8195215 0.86 ACACB (0.35) SMN1; SMN2CTSBACACBMEN1KMT2A
SCHEMBL12943109 0.85 ACACB (0.35) SMN1; SMN2ACACBMEN1KMT2AGAA
SCHEMBL12943110 0.84 CTSD (0.34) ACACBMEN1KMT2AGAACYP2D6
SCHEMBL12943104 0.81 IL1RN (0.33)
SCHEMBL12943212 0.78 CTSB (0.37) CTSBACACBALDH1A1
SCHEMBL8208994 0.78 MME (0.42) MMP1MMP2MMP9ALDH1A1
SCHEMBL8202825 0.78 PTPN1 (0.44) MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008048121-A2 MACROCYCLIC CYSTEINE PROTEASE INHIBITORS AND COMPOSITIONS THEREOF LINCOLN UNIVERSITY (NZ) 2008-04-24 WO disclosed