Protizinic Acid

Protizinic Acid

SCHEMBL8208239

COc1ccc2c(c1)Sc1ccc(C(C)C(=O)O)cc1N2C.O=C(O)c1ccccc1O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHE

The experimentally established mechanism targets of Protizinic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.44
AKR1C2 P52895 4/20 0.44
PTGS2 P35354 3/20 0.44
PTGS1 P23219 2/20 0.44
CYP1A2 P05177 2/20 0.44
CDC42 P60953 1/20 0.44
RAC1 P63000 1/20 0.44
TSHR P16473 1/20 0.44
SLC22A6 Q4U2R8 1/20 0.44
KDM4E B2RXH2 3/20 0.43
TP53 P04637 2/20 0.43
MAPK1 P28482 2/20 0.43
SNCA P37840 4/20 0.42
HPGD P15428 2/20 0.41
ALOX15 P16050 2/20 0.41
CYP2C19 P33261 2/20 0.41
LMNA P02545 2/20 0.41
PGR P06401 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Protizinic Acid SCHEMBL29359535 0.89 AKR1C3 (0.54) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
Protizinic Acid SCHEMBL18309842 0.89 AKR1C3 (0.54) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
Protizinic Acid SCHEMBL25022 0.89 AKR1C3 (0.54) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
Naproxen SCHEMBL27586482 0.78 AKR1C3 (0.72) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
Naproxen SCHEMBL2038673 0.78 AKR1C3 (0.72) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
SCHEMBL10618628 0.78 NOX1 (0.58) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
SCHEMBL2739325 0.76 SNCA (0.59) PTGS1CYP1A2KDM4ETP53MAPK1
Protizinic Acid SCHEMBL2072946 0.73 PTGS1 (0.63) AKR1C3AKR1C2PTGS2PTGS1CYP1A2
SCHEMBL11255517 0.73 SNCA (0.53) PTGS1CYP1A2KDM4ETP53MAPK1
Rosmarinic Acid SCHEMBL9446582 0.72 MMP1 (0.56) CYP1A2KDM4ESNCAHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977725-A1 NEW FATTY ACID DERIVATIVES NORSK HYDRO ASA (NO) 2000-02-09 EP disclosed
WO-1998032718-A1 NEW FATTY ACID DERIVATIVES NORSK HYDRO ASA (NO) 1998-07-30 WO disclosed