SCHEMBL8209631

SCHEMBL8209631

NC(=O)N1C(=O)[C@H](c2ccc(OCc3ccc(F)cc3)cc2)C[C@@H]1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 1/20 0.51
NPC1 O15118 1/20 0.51
POLB P06746 1/20 0.51
RAB9A P51151 1/20 0.51
MAOB P27338 11/20 0.50
KCNH2 Q12809 1/20 0.50
PARP10 Q53GL7 1/20 0.50
NR4A2 P43354 1/20 0.48
HRH3 Q9Y5N1 1/20 0.46
KDM1A O60341 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
MAOA P21397 4/20 0.41
GSK3B P49841 1/20 0.41
BACE1 P56817 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208997 0.90 MAOB (0.42) S1PR5NPC1POLBRAB9AMAOB
SCHEMBL8209192 0.90 MMP13 (0.49) S1PR5NPC1RAB9AMAOBKCNH2
SCHEMBL8213085 0.87 MMP13 (0.46) NPC1POLBRAB9AKCNH2PARP10
SCHEMBL8212956 0.83 MMP13 (0.42) POLBMAOBKDM1A
SCHEMBL8209442 0.77 KDM1A (0.43) NPC1RAB9AKCNH2PARP10KDM1A
SCHEMBL8210831 0.74 BTK (0.35) MAOBKCNH2KDM1AMAOA
SCHEMBL19609293 0.73 CYP4F2 (0.57) S1PR5MAOBKCNH2PARP10NR4A2
SCHEMBL8208991 0.73 NPC1 (0.41) NPC1RAB9AMAOBKDM1AMAOA
SCHEMBL8211740 0.72 ROCK2 (0.38)
SCHEMBL28648433 0.71 MAOB (0.56) S1PR5NPC1POLBRAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114361-A INHIBITORS OF MATRIX METALLOPROTEINASES AND REPROLYSIN; ADMINISTERING TO TREAT CONDITIONS WHICH CAN BE TREATED BY THE INHIBITION OF THESE ENZYMES PFIZER INC. (US) 2000-09-05 US claimed