SCHEMBL8209747

SCHEMBL8209747

CC(Sc1c2ccccc2nc2ccccc12)Sc1c2ccccc2nc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.46
POLB P06746 2/20 0.45
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 4/20 0.45
HPGD P15428 3/20 0.45
MAOA P21397 2/20 0.45
GLA P06280 2/20 0.45
CASP1 P29466 2/20 0.45
CASP7 P55210 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HSD17B10 Q99714 2/20 0.45
CHRM2 P08172 1/20 0.45
ADRA2A P08913 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CHRM1 P11229 1/20 0.45
NQO2 P16083 1/20 0.45
DRD1 P21728 1/20 0.45
ACHE P22303 1/20 0.45
SLC6A2 P23975 1/20 0.45
ADRA1A P35348 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212730 0.85 KDM1A (0.50) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL8207048 0.79 ALDH1A1 (0.47) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL17423359 0.76 KDM4E (0.50) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL17423904 0.71 KDM4E (0.50) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL1102408 0.71 KDM4E (0.50) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL7869236 0.70 KDM1A (0.48) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL3344226 0.68 POLB (0.63) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL3347479 0.68 POLB (0.47) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL3349467 0.68 MAOA (0.52) KDM1APOLBALDH1A1KDM4EHPGD
SCHEMBL31678400 0.67 GPR3 (0.58) KDM1APOLBALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979078-A4 SUBSTITUTED BIS-ACRIDINES AND RELATED COMPOUNDS AS CCR5 RECEPTOR LIGANDS, ANTI-INFLAMMATORY AGENTS AND ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2000-06-21 EP claimed
EP-0979078-A1 SUBSTITUTED BIS-ACRIDINES AND RELATED COMPOUNDS AS CCR5 RECEPTOR LIGANDS, ANTI-INFLAMMATORY AGENTS AND ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-16 EP claimed
WO-1998030218-A1 SUBSTITUTED BIS-ACRIDINES AND RELATED COMPOUNDS AS CCR5 RECEPTOR LIGANDS, ANTI-INFLAMMATORY AGENTS AND ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 1998-07-16 WO claimed