SCHEMBL8209788

SCHEMBL8209788

CC(c1cn(C(=O)c2ccccc2Cl)c2ccc(OC3CCCCC3)cc12)C1CCCN1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE4B Q07343 1/20 0.37
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
HIF1A Q16665 1/20 0.34
HRH1 P35367 1/20 0.33
CCR3 P51677 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
MAOB P27338 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
SLC6A3 Q01959 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8211654 0.91 PTGS1 (0.35) KMT2APTGS1PTGS2HIF1AHRH3
SCHEMBL8201991 0.89 HIF1A (0.41) ALDH1A1KMT2APDE4BPTGS1PTGS2
SCHEMBL8213329 0.88 PTGS1 (0.38) ALDH1A1PTGS1PTGS2MAOBSLC6A3
SCHEMBL8209083 0.84 PDE4B (0.38) ALDH1A1KMT2APDE4BPTGS1PTGS2
SCHEMBL8201465 0.76 HTR6 (0.43)
SCHEMBL8209787 0.75 SLC6A2 (0.40) MAPTKMT2APTGS2SLC6A3SLC6A2
SCHEMBL8201598 0.74 AKR1C3 (0.46) KMT2APTGS1
SCHEMBL8208559 0.73 KMT2A (0.51) ALDH1A1KMT2ACNR2
SCHEMBL8209786 0.73 HTR6 (0.52) ALDH1A1MAPTKMT2APDE4BHRH3
SCHEMBL8209783 0.73 HTR6 (0.52) ALDH1A1MAPTKMT2APDE4BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US claimed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO claimed
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US disclosed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO disclosed