SCHEMBL8213329

SCHEMBL8213329

CC(c1cn(C(=O)c2ccccc2)c2ccc(OC3CCCCC3)cc12)C1CCCN1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
HTR6 P50406 1/20 0.38
EGLN1 Q9GZT9 1/20 0.35
ACHE P22303 1/20 0.35
MAOB P27338 2/20 0.35
MAOA P21397 1/20 0.35
SLC6A3 Q01959 5/20 0.35
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 2/20 0.35
DHFR P00374 1/20 0.35
APP P05067 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8209083 0.92 PDE4B (0.38) PTGS1PTGS2HTR6SLC6A3SLC6A2
SCHEMBL8209788 0.88 ALDH1A1 (0.38) PTGS1PTGS2MAOBSLC6A3SLC6A2
SCHEMBL8201991 0.88 HIF1A (0.41) PTGS1PTGS2ALDH1A1
SCHEMBL8211654 0.87 PTGS1 (0.35) PTGS1PTGS2SLC6A3SLC6A2SLC6A4
SCHEMBL8209787 0.83 SLC6A2 (0.40) PTGS2HTR6SLC6A3SLC6A2SLC6A4
SCHEMBL6968879 0.83 DYRK1A (0.42) HTR6SLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL8208589 0.83 KMT2A (0.44) PTGS2HTR6SLC6A3SLC6A2SLC6A4
SCHEMBL8201465 0.81 HTR6 (0.43) HTR6
SCHEMBL8208559 0.80 KMT2A (0.51) HTR6ACHEALDH1A1
SCHEMBL8201598 0.79 AKR1C3 (0.46) PTGS1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US claimed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO claimed
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US disclosed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO disclosed