SCHEMBL8201598

SCHEMBL8201598

COc1ccc(C(=O)n2cc(C(C)C3CCCN3)c3cc(Cl)ccc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 11/20 0.46
AKR1C2 P52895 8/20 0.46
PTGS1 P23219 2/20 0.46
AKR1C4 P17516 1/20 0.46
AR P10275 1/20 0.40
KMT2A Q03164 1/20 0.39
MGLL Q99685 1/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8208574 0.89 AKR1C3 (0.42) AKR1C3AKR1C2KMT2AMGLL
SCHEMBL8209787 0.89 SLC6A2 (0.40) KMT2A
SCHEMBL8208559 0.87 KMT2A (0.51) KMT2AACHE
SCHEMBL8209083 0.87 PDE4B (0.38) AKR1C3AKR1C2PTGS1AKR1C4KMT2A
SCHEMBL8201582 0.80 HTR6 (0.50)
SCHEMBL8213329 0.79 PTGS1 (0.38) PTGS1ACHE
SCHEMBL6968879 0.77 DYRK1A (0.42) KMT2A
SCHEMBL8208589 0.76 KMT2A (0.44) KMT2A
SCHEMBL8200926 0.75 KMT2A (0.47) KMT2AACHE
SCHEMBL8211654 0.75 PTGS1 (0.35) PTGS1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US claimed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO claimed
US-6100291-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ALLELIX BIOPHARMACEUTICALS INC. (CA) 2000-08-08 US disclosed
WO-1999047516-A1 3-(2-PYRROLIDINYLMETHYL)-INDOLE COMPOUNDS HAVING 5-HT6 AFFINITY SLASSI ABDELMALIK (CA) 1999-09-23 WO disclosed