SCHEMBL8212932

SCHEMBL8212932

CON(C)C(=O)[C@@H]1C[C@@H](OS(C)(=O)=O)CN1C(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.42
MMP2 P08253 1/20 0.37
ANPEP P15144 1/20 0.37
NR1H2 P55055 3/20 0.33
NR1H3 Q13133 2/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD11B1 P28845 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
MCL1 Q07820 4/20 0.32
GPR119 Q8TDV5 1/20 0.31
PTPN1 P18031 1/20 0.31
USP30 Q70CQ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18538108 0.86 UCHL1 (0.53) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL30501862 0.86 UCHL1 (0.53) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL27393752 0.86 UCHL1 (0.53) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL25619159 0.86 UCHL1 (0.53) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL31340923 0.86 UCHL1 (0.53) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL18577225 0.85 UCHL1 (0.45) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL18577227 0.85 UCHL1 (0.45) UCHL1NR1H2CYP1A2POLBCYP3A4
SCHEMBL7805563 0.83 MMP2 (0.48) UCHL1MMP2ANPEPNR1H2NR1H3
SCHEMBL5691732 0.83 MMP2 (0.48) UCHL1MMP2ANPEPNR1H2NR1H3
SCHEMBL489252 0.83 MMP2 (0.48) UCHL1MMP2ANPEPNR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054865-A1 FARNESYL TRANSFERASE INHIBITORS AstraZeneca UK Limited (GB) 2000-11-29 EP disclosed
WO-1999041235-A1 FARNESYL TRANSFERASE INHIBITORS ASTRAZENECA UK LIMITED (GB) 1999-08-19 WO disclosed