SCHEMBL8212957

SCHEMBL8212957

[c]1ccc2c(c1-c1ccccc1)OCO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP1B1 Q16678 2/20 0.39
CYP1A1 P04798 1/20 0.39
PTGS2 P35354 3/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
PKM P14618 2/20 0.33
MEN1 O00255 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
TSHR P16473 1/20 0.32
BAD Q92934 1/20 0.32
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL161183 0.85 ABCG2 (0.39) ABCG2PKMTSHRBADTXNRD1
SCHEMBL8638641 0.83 MAPT (0.39) PTGS2MEN1NPC1RAB9AKMT2A
SCHEMBL9740282 0.83 RIPK3 (0.37) KDM4EMAPT
SCHEMBL9738660 0.79 KDM4E (0.41) PTGS2MEN1NPC1RAB9AKMT2A
SCHEMBL6784931 0.78 HSP90AA1 (0.30)
SCHEMBL11571390 0.75 PREP (0.43) PTGS2PKMMEN1NPC1RAB9A
SCHEMBL8925096 0.72 ABCG2 (0.38) ABCG2PTGS2HTR1ADRD2MEN1
SCHEMBL6210971 0.72 PDE4A (0.41) MEN1NPC1RAB9AKMT2ATSHR
SCHEMBL15377351 0.72 ALOX5 (0.45) PTGS2MEN1NPC1RAB9AKMT2A
SCHEMBL3404505 0.71 ABCG2 (0.37) ABCG2PTGS2TXNRD1TXNRD3TXNRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6030975-A ANTAGONIST OF ENDOTHELINS, I.E. INHIBITION OF BINDING WITH RECEPTOR; ANTITUMOR AND -CARCINOGENIC AGENTS; SIDE EFFECT REDUCTION BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed