SCHEMBL8213312

SCHEMBL8213312

O=C(C1CC1c1ccc2ccccc2n1)C12CC3CCCC(C1)C(C3)C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM5 Q9NZQ8 1/20 0.37
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
OPRK1 P41145 1/20 0.33
HSD11B1 P28845 3/20 0.33
CNR1 P21554 1/20 0.33
KDM2B Q8NHM5 2/20 0.32
MGAM O43451 1/20 0.32
F2R P25116 1/20 0.32
GRM1 Q13255 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4731571 0.85 CNR1 (0.43) TRPM5ALDH1A1NPC1RAB9AMEN1
SCHEMBL8215059 0.81 GRM1 (0.40) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL8215134 0.72 ITK (0.35) ALDH1A1NPC1RAB9AMEN1MAPT
SCHEMBL2136784 0.71 MGAM (0.50) TRPM5ALDH1A1NPC1RAB9AMEN1
SCHEMBL2136780 0.71 MGAM (0.50) TRPM5ALDH1A1NPC1RAB9AMEN1
SCHEMBL8219547 0.70 CNR2 (0.35) ALDH1A1NPC1RAB9AMEN1MAPT
SCHEMBL6085541 0.70 HSD11B1 (0.44) ALDH1A1NPC1RAB9AMEN1TP53
SCHEMBL8215561 0.70 HSD11B1 (0.45) ALDH1A1RAB9AMEN1CYP3A4MAPT
SCHEMBL8212845 0.68 ALDH1A1 (0.42) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL8211978 0.68 GRM1 (0.40) GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed