SCHEMBL8212845

SCHEMBL8212845

COc1ccc2ncc(C3CC3C(=O)C34CC5CCCC(C3)C(C5)C4)cc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
F2 P00734 1/20 0.42
GLA P06280 1/20 0.42
HPGD P15428 1/20 0.42
AURKA O14965 1/20 0.40
LCK P06239 1/20 0.40
FYN P06241 1/20 0.40
IGF1R P08069 1/20 0.40
MET P08581 1/20 0.40
KIT P10721 1/20 0.40
FGFR2 P21802 1/20 0.40
EPHA2 P29317 1/20 0.40
LTK P29376 1/20 0.40
AXL P30530 1/20 0.40
FLT3 P36888 1/20 0.40
MST1R Q04912 1/20 0.40
ITK Q08881 5/20 0.38
GRM1 Q13255 1/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8215082 0.93 HPGDS (0.42) HPGDS
SCHEMBL4729426 0.88 ALDH1A1 (0.49) ALDH1A1F2GLAHPGDAURKA
SCHEMBL8213684 0.87 PDGFRB (0.46) GRM1PDGFRBPDGFRA
SCHEMBL8215059 0.85 GRM1 (0.40) ALDH1A1GRM1NPC1RAB9AMEN1
SCHEMBL8211978 0.81 GRM1 (0.40) GRM1
SCHEMBL4728861 0.80 HPGDS (0.46) ITKGRM1HPGDS
SCHEMBL8215134 0.79 ITK (0.35) ALDH1A1HPGDITKGRM1HSD11B1
SCHEMBL8215665 0.75 RXRA (0.36) ALDH1A1GRM1NPC1
SCHEMBL4729407 0.74 PDGFRB (0.48) ALDH1A1GRM1MEN1KMT2APDGFRB
SCHEMBL8219547 0.72 CNR2 (0.35) ALDH1A1HPGDGRM1HSD11B1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed