SCHEMBL4731571

SCHEMBL4731571

O=C(C1CC1c1ccc2ccccc2n1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.43
TRPM5 Q9NZQ8 1/20 0.42
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
LMNA P02545 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
HTT P42858 2/20 0.41
GRM1 Q13255 1/20 0.41
MAPK1 P28482 3/20 0.40
CYP3A4 P08684 2/20 0.39
MGAM O43451 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8213312 0.85 TRPM5 (0.37) CNR1TRPM5MAPTSMN1; SMN2NPC1
SCHEMBL2136784 0.79 MGAM (0.50) TRPM5MAPTKDM4ESMN1; SMN2LMNA
SCHEMBL2136780 0.79 MGAM (0.50) TRPM5MAPTKDM4ESMN1; SMN2LMNA
SCHEMBL4731345 0.77 P2RX7 (0.49) MAPTKDM4ELMNARAB9AHTT
SCHEMBL4728893 0.76 GRM1 (0.51) CNR1MAPTKDM4ESMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL4728933 0.76 P2RX7 (0.48) MAPTKDM4ELMNARAB9AHTT
Hydrochloric Acid SCHEMBL4727017 0.75 GRM1 (0.50) CNR1MAPTKDM4ESMN1; SMN2LMNA
SCHEMBL16278329 0.74 TRPM5 (0.44) TRPM5MAPTKDM4ESMN1; SMN2NPC1
SCHEMBL16278689 0.74 TRPM5 (0.54) TRPM5MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL16283865 0.74 TRPM5 (0.44) TRPM5MAPTKDM4ESMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed