SCHEMBL8217795

SCHEMBL8217795

O=c1cc(Cl)n(Cc2ccccc2I)c(=O)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
HPGD P15428 3/20 0.47
CYP3A4 P08684 1/20 0.47
KMT2A Q03164 6/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
DPP4 P27487 2/20 0.37
TSHR P16473 1/20 0.36
PGR P06401 1/20 0.36
MEN1 O00255 4/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
HTR2C P28335 1/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8219650 0.82 DPP4 (0.53) ALDH1A1HPGDCYP3A4KMT2AL3MBTL1
SCHEMBL25130124 0.81 HPGD (0.68) ALDH1A1HPGDCYP3A4KMT2AL3MBTL1
SCHEMBL390246 0.79 DPP4 (0.56) ALDH1A1HPGDCYP3A4KMT2ADPP4
SCHEMBL8217925 0.75 HSP90AA1 (0.41) ALDH1A1HPGDCYP3A4KMT2AMAPT
SCHEMBL10048200 0.73 LMNA (0.54) ALDH1A1HPGDCYP3A4KMT2AL3MBTL1
SCHEMBL30753174 0.73 TRAP1 (0.40) ALDH1A1HPGDCYP3A4KMT2AL3MBTL1
SCHEMBL8216227 0.72 ALDH1A1 (0.48) ALDH1A1HPGDCYP3A4KMT2AL3MBTL1
SCHEMBL8216928 0.72 KMT2A (0.44) ALDH1A1HPGDCYP3A4KMT2AMAPT
SCHEMBL18931749 0.71 KMT2A (0.50) ALDH1A1HPGDCYP3A4KMT2AL3MBTL1
SCHEMBL13206724 0.70 KMT2A (0.43) ALDH1A1HPGDCYP3A4KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188275-B2 hydrolase enzyme inhibors such as 2-(6-Chloro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethyl)-benzonitrile TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-05-29 US claimed