SCHEMBL8219650

SCHEMBL8219650

O=c1cc(Cl)n(Cc2ccccc2Br)c(=O)[nH]1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.53
HPGD P15428 3/20 0.47
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
TSHR P16473 1/20 0.36
PGR P06401 1/20 0.36
MEN1 O00255 1/20 0.36
CYP2A13 Q16696 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8217795 0.82 ALDH1A1 (0.47) DPP4HPGDALDH1A1CYP3A4KMT2A
SCHEMBL8215220 0.82 KMT2A (0.43) DPP4HPGDALDH1A1CYP3A4KMT2A
SCHEMBL25130124 0.81 HPGD (0.68) HPGDALDH1A1CYP3A4KMT2AL3MBTL1
SCHEMBL390246 0.79 DPP4 (0.56) DPP4HPGDALDH1A1CYP3A4KMT2A
SCHEMBL8220301 0.75 DPP4 (0.54) DPP4HPGDALDH1A1CYP3A4CYP1A2
SCHEMBL8217925 0.75 HSP90AA1 (0.41) DPP4HPGDALDH1A1CYP3A4KMT2A
SCHEMBL10048200 0.73 LMNA (0.54) HPGDALDH1A1CYP3A4KMT2AL3MBTL1
SCHEMBL4211224 0.73 CA12 (0.50) DPP4HPGDALDH1A1CYP1A2CYP2D6
SCHEMBL30753174 0.73 TRAP1 (0.40) HPGDALDH1A1CYP3A4CYP1A2CYP2D6
SCHEMBL8216227 0.72 ALDH1A1 (0.48) DPP4HPGDALDH1A1CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188275-B2 hydrolase enzyme inhibors such as 2-(6-Chloro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethyl)-benzonitrile TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-05-29 US claimed