SCHEMBL8218521

SCHEMBL8218521

CC(C)C[C@H]1COc2ccsc2C(N)=N1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.70
NOS2 P35228 4/20 0.70
NOS1 P29475 3/20 0.70
TAAR1 Q96RJ0 4/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP2D6 P10635 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195096 0.85 NOS2 (0.80) NOS3NOS2NOS1TAAR1CYP2D6
SCHEMBL8214849 0.82 NOS3 (1.00) NOS3NOS2NOS1TAAR1
SCHEMBL8186392 0.80 NOS2 (0.85) NOS3NOS2NOS1TAAR1
SCHEMBL8206872 0.77 NOS2 (0.64) NOS3NOS2NOS1TAAR1
SCHEMBL8208391 0.69 NOS2 (0.59) NOS3NOS2NOS1TAAR1NPC1
SCHEMBL11818478 0.69 TAAR1 (0.61) TAAR1CYP2D6
SCHEMBL21067657 0.66 NOS3 (0.93) NOS3NOS2NOS1TAAR1
SCHEMBL4946193 0.64 NPC1 (0.42) NOS3NOS2NOS1TAAR1NPC1
SCHEMBL28738590 0.64 NPC1 (0.42) NOS3NOS2NOS1TAAR1NPC1
SCHEMBL23249399 0.62 NPC1 (0.41) NOS3NOS2NOS1TAAR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO claimed
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO disclosed