SCHEMBL8218893

SCHEMBL8218893

N#CN=C(NCCOCCOC(c1ccc(F)cc1)c1ccc(F)cc1)Nc1ccncc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.37
IKBKB O14920 1/20 0.37
SLC6A2 P23975 7/20 0.37
SLC6A4 P31645 7/20 0.37
SLC6A3 Q01959 7/20 0.37
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TAAR1 Q96RJ0 1/20 0.34
CYP3A4 P08684 4/20 0.32
CYP2C9 P11712 3/20 0.32
CYP2C19 P33261 3/20 0.32
CYP1A2 P05177 2/20 0.32
NFKB1 P19838 2/20 0.32
MAPK1 P28482 2/20 0.32
HIF1A Q16665 2/20 0.32
LMNA P02545 2/20 0.32
BLM P54132 2/20 0.32
PMP22 Q01453 2/20 0.32
CYP2D6 P10635 2/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196335 0.90 LMNA (0.38) NAMPTIKBKBCYP3A4CYP2C9CYP2C19
SCHEMBL7982467 0.80 SLC6A2 (0.37) NAMPTSLC6A2SLC6A4SLC6A3MEN1
SCHEMBL7982471 0.80 SLC6A2 (0.37) NAMPTSLC6A2SLC6A4SLC6A3MEN1
SCHEMBL8198968 0.79 IKBKB (0.44) NAMPTIKBKBKMT2ACYP3A4CYP2C9
SCHEMBL8199078 0.78 HTR1A (0.42) NAMPTIKBKBSLC6A2SLC6A4SLC6A3
SCHEMBL8195688 0.78 IKBKB (0.43) NAMPTIKBKBKMT2ACYP3A4CYP2C9
SCHEMBL8195918 0.76 IKBKB (0.37) NAMPTIKBKBCYP3A4CYP2C9CYP2C19
SCHEMBL8195627 0.75 IKBKB (0.46) NAMPTIKBKBMEN1KMT2ACYP3A4
SCHEMBL8195516 0.74 IKBKB (0.63) NAMPTIKBKBMEN1KMT2ACYP3A4
SCHEMBL8200614 0.71 IKBKB (0.38) NAMPTIKBKBMEN1KMT2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO disclosed