SCHEMBL8219487

SCHEMBL8219487

N=C(S)S(=O)(=O)Cc1cc(N)nc(-c2ccc(NC(=O)NC3CC3)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.40
MTOR P42345 6/20 0.40
PIK3CD O00329 4/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
RAB9A P51151 2/20 0.39
KLKB1 P03952 1/20 0.39
EPHX1 P07099 1/20 0.39
GAA P10253 1/20 0.39
EPHX2 P34913 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
KIT P10721 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8212640 0.87 PIK3CA (0.51) PIK3CAMTORPIK3CDCA12CA1
SCHEMBL8217170 0.86 PIK3CA (0.42) PIK3CAMTORPIK3CDKDM4EMEN1
SCHEMBL8219567 0.83 PIK3CA (0.42) PIK3CAMTORPIK3CDCA12CA1
SCHEMBL8205208 0.83 PIK3CA (0.42) PIK3CAMTORPIK3CDCA12CA1
SCHEMBL8212559 0.83 MEN1 (0.46) PIK3CAMTORPIK3CDCA12CA1
SCHEMBL8206186 0.82 RAB9A (0.45) PIK3CAMTORPIK3CDCA12CA1
SCHEMBL8218892 0.81 PIK3CA (0.48) PIK3CAMTORCA12CA1CA2
SCHEMBL8213009 0.81 PIK3CA (0.56) PIK3CAMTORPIK3CDCA12CA1
SCHEMBL8213961 0.81 CA12 (0.47) CA12CA1CA2CA9RAB9A
SCHEMBL8214242 0.80 CYP3A4 (0.44) PIK3CAMTORPIK3CDCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008023159-A1 MORPHOLINO PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF PROLIFERATIVE DISORDERS ASTRAZENECA AB (SE) 2008-02-28 WO disclosed