SCHEMBL8220530

SCHEMBL8220530

CCP(=O)(CC)Cc1ccc(C(N)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.47
PLA2G2A P14555 1/20 0.47
PARP10 Q53GL7 7/20 0.46
EPHX2 P34913 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
HDAC1 Q13547 1/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PARP4 Q9UKK3 2/20 0.41
PARP1 P09874 2/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
CYP17A1 P05093 1/20 0.41
MAPK1 P28482 2/20 0.40
APAF1 O14727 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28741620 0.83 ALDH1A1 (0.59) EPHX2NR1H4KMT2AMEN1SMN1; SMN2
SCHEMBL4663159 0.79 LOXL2 (0.56) KMT2AMEN1SMN1; SMN2KDM4ENPC1
SCHEMBL5276387 0.77 PARP10 (0.50) PLA2G10PLA2G2APARP10EPHX2NR1H4
SCHEMBL10910029 0.76 ESR1 (0.42) KDM4ECA2ALDH1A1CYP3A4HSD17B10
SCHEMBL2033357 0.76 FDPS (0.42) HDAC1MAPK1ALDH1A1MAOBCYP3A4
SCHEMBL3249156 0.76 HRH3 (0.43) HDAC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL178439 0.76 ALDH1A1 (0.64) PLA2G10PLA2G2APARP10EPHX2NR1H4
SCHEMBL2464783 0.72 PLK1 (0.60) PLA2G10PLA2G2APARP10KMT2AKDM4E
SCHEMBL28151928 0.72 PLA2G10 (0.53) PLA2G10PLA2G2APARP10EPHX2NR1H4
SCHEMBL7809399 0.72 HDAC8 (0.64) PLA2G10PLA2G2APARP10PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008010985-A2 PHOSPHORUS DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2008-01-24 WO disclosed