SCHEMBL8239148

SCHEMBL8239148

CC(C)(C)OC(=O)N[C@@H](CCc1ccc(C(C)(C)C)cc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.57
CTSS P25774 5/20 0.57
PPARA Q07869 10/20 0.52
PPARG P37231 9/20 0.52
PPARD Q03181 2/20 0.50
TGM2 P21980 1/20 0.49
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
ACE P12821 1/20 0.48
CA2 P00918 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12305805 1.00 CTSK (0.57) CTSKCTSSPPARAPPARGPPARD
SCHEMBL12475131 0.90 PPARA (0.64) CTSKCTSSPPARAPPARGPPARD
SCHEMBL12475133 0.90 PPARA (0.64) CTSKCTSSPPARAPPARGPPARD
SCHEMBL31407637 0.90 PPARA (0.64) CTSKCTSSPPARAPPARGPPARD
SCHEMBL23705756 0.88 CTSK (0.58) CTSKCTSSPPARAPPARGPPARD
SCHEMBL21409154 0.88 PPARA (0.62) CTSKCTSSPPARAPPARGPPARD
SCHEMBL12305799 0.88 PPARA (0.62) CTSKCTSSPPARAPPARGPPARD
SCHEMBL8316046 0.88 CTSK (0.58) CTSKCTSSPPARAPPARGPPARD
SCHEMBL3773563 0.88 CTSK (0.58) CTSKCTSSPPARAPPARGPPARD
SCHEMBL12305804 0.88 CTSK (0.58) CTSKCTSSPPARAPPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8338471-B2 (2,5-dioxoimidazolidin-i-yl)-n-hydroxy-acetamides as metalloproteinase inhibitors MEDIVIR AB (SE) 2012-12-25 US disclosed
US-20120015994-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MEDIVIR AB (SE) 2012-01-19 US disclosed
WO-2007068474-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MEDIVIR AB (SE) 2007-06-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120015994-A1 (2,5-DIOXOIMIDAZOLIDIN-I-YL)-N-HYDROXY-ACETAMIDES AS METALLOPROTEINASE INHIBITORS MMP12, MMP13, MMP14 CTSK 417/4885CTSS 186/4885PPARA 1865/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.