SCHEMBL8239647

SCHEMBL8239647

Cc1ccc(N2CC=CCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.48
MAPT P10636 6/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
AKR1C3 P42330 1/20 0.39
POLB P06746 1/20 0.37
HTR7 P34969 1/20 0.37
CRHR1 P34998 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
DHFR P00374 1/20 0.36
PKM P14618 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5854414 0.87 ADRB1 (0.54) ADRB1MAPTNPSR1MEN1KMT2A
SCHEMBL4071866 0.81 ADRB1 (0.50) ADRB1MAPTNPSR1MEN1KMT2A
SCHEMBL1889513 0.80 LMNA (0.46) ADRB1MAPTMEN1KMT2APOLB
SCHEMBL5276484 0.79 SIGMAR1 (0.48) ADRB1MAPTNPSR1KMT2AAKR1C3
SCHEMBL4317647 0.79 MAPT (0.50) MAPTNPSR1MEN1KMT2APOLB
SCHEMBL4565389 0.79 MAPK1 (0.48) MAPTNPSR1MEN1KMT2APOLB
SCHEMBL8263647 0.79 ADRB1 (0.56) ADRB1MAPTHTR7RAB9ADHFR
SCHEMBL13105671 0.79 IKBKB (0.41) MAPTNPSR1MEN1KMT2AHTR7
SCHEMBL26814948 0.79 ALDH1A1 (0.40) MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL7038234 0.79 ADRB1 (0.53) ADRB1MAPTMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007089768-A2 4-ARYL-2-AMINO-PYRIMIDINES OR 4-ARYL-2-AMINOALKYL-PYRIMIDINES AS JAK-2 MODULATORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM EXELIXIS, INC. (US) 2007-08-09 WO disclosed