SCHEMBL8239706

SCHEMBL8239706

O=C(O)c1ccc(Oc2ncccc2C(=O)N2CCN(c3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 2/20 0.43
CYP3A4 P08684 1/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD11B1 P28845 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ENPP2 Q13822 2/20 0.42
SLC6A7 Q99884 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
TRPA1 O75762 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
KMT2A Q03164 1/20 0.41
NOTUM Q6P988 3/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8245894 0.89 POLB (0.47) POLBSMN1; SMN2MAPTHTTENPP2
SCHEMBL4761009 0.85 MEN1 (0.56) POLBSMN1; SMN2MAPTCYP3A4GAA
SCHEMBL4762716 0.85 SMN1; SMN2 (0.51) POLBSMN1; SMN2MAPTCYP3A4GAA
SCHEMBL4762664 0.84 POLB (0.56) POLBMAPTENPP2SLC6A7MEN1
SCHEMBL4761369 0.84 POLB (0.52) POLBMAPTENPP2SLC6A7MEN1
SCHEMBL4762542 0.83 HSD11B1 (0.53) SMN1; SMN2MAPTCYP3A4GAACYP2C9
SCHEMBL4763187 0.82 SMN1; SMN2 (0.55) SMN1; SMN2MAPTHTTKDM4ESLC6A7
SCHEMBL4764201 0.81 POLB (0.49) POLBMAPTGAAKDM4ESLC6A7
SCHEMBL4761689 0.81 POLB (0.52) POLBMAPTGAANPSR1KDM4E
SCHEMBL8246475 0.81 ALDH1A1 (0.58) POLBSMN1; SMN2MAPTGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007009635-A1 PHENYL SUBSTITUTED PIPERAZINE-DERIVATIVES AS INHIBITORS OF PLAMINOGENIC ACTIVATOR INHIBITORS-I (PAI-I) BAYER HEALTHCARE AG (DE) 2007-01-25 WO disclosed