SCHEMBL8247665

SCHEMBL8247665

Nc1cccc(CCCC2CCN(Cc3cc(Cl)c4c(c3)CN(CC3CC3)C4=O)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.49
PARP2 Q9UGN5 2/20 0.46
ACHE P22303 6/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1002789 0.87 PARP1 (0.45) PARP1PARP2ACHE
SCHEMBL2024915 0.76 PARP1 (0.43) PARP1PARP2ACHE
SCHEMBL2023586 0.74 PARP1 (0.46) PARP1PARP2ACHE
SCHEMBL1002428 0.72 PARP1 (0.44) PARP1PARP2
SCHEMBL8271635 0.71 PARP1 (0.39) PARP1PARP2ACHE
SCHEMBL8240044 0.71 ALDH1A1 (0.47) PARP1PARP2ACHE
SCHEMBL12641815 0.70 ACHE (0.46) PARP1PARP2ACHE
SCHEMBL17064545 0.69 MAOA (0.53)
SCHEMBL8240048 0.69 PARP1 (0.41) PARP1PARP2ACHE
SCHEMBL2024499 0.69 PARP1 (0.39) PARP1PARP2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007021309-A1 SUBSTITUTED ISOINDOLONES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2007-02-22 WO disclosed
WO-2006020879-A1 ISOINDOLONE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2006-02-23 WO disclosed